The preparation of 1,2,3-trisubstituted guanidines

Alan R. Katritzky; Niveen M. Khashab; Sergey Bobrov

doi:10.1002/hlca.200590131

The preparation of 1,2,3-trisubstituted guanidines

Alan R. Katritzky^*, Niveen M. Khashab, Sergey Bobrov

^*Corresponding author for this work

Research output: Contribution to journal › Article › peer-review

28 Scopus citations

Abstract

An operationally straightforward and efficient benzotriazole-based method for the guanylation of diverse amines by use of the new reagent classes (bis-benzotriazol-1-yl-methylene)amines 13a-13f and benzotriazole-1- carboxamidines 17a-17i is described. The preparation is described for a variety of both acyclic and cyclic 1,2,3-trisubstituted guanidines in high yields.

Original language	English (US)
Pages (from-to)	1664-1675
Number of pages	12
Journal	Helvetica Chimica Acta
Volume	88
Issue number	7
DOIs	https://doi.org/10.1002/hlca.200590131
State	Published - 2005
Externally published	Yes

ASJC Scopus subject areas

Catalysis
Biochemistry
Drug Discovery
Physical and Theoretical Chemistry
Organic Chemistry
Inorganic Chemistry

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10.1002/hlca.200590131

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abstract = "An operationally straightforward and efficient benzotriazole-based method for the guanylation of diverse amines by use of the new reagent classes (bis-benzotriazol-1-yl-methylene)amines 13a-13f and benzotriazole-1- carboxamidines 17a-17i is described. The preparation is described for a variety of both acyclic and cyclic 1,2,3-trisubstituted guanidines in high yields.",

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AU - Bobrov, Sergey

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AB - An operationally straightforward and efficient benzotriazole-based method for the guanylation of diverse amines by use of the new reagent classes (bis-benzotriazol-1-yl-methylene)amines 13a-13f and benzotriazole-1- carboxamidines 17a-17i is described. The preparation is described for a variety of both acyclic and cyclic 1,2,3-trisubstituted guanidines in high yields.

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M3 - Article

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ER -

The preparation of 1,2,3-trisubstituted guanidines

Abstract

ASJC Scopus subject areas

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